doi: 10.1016/s0960-894x(00)00558-8.
Solid-phase synthesis of 2,3-disubstituted indoles: discovery of a novel, high-affinity, selective h5-HT2A antagonist
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- PMID: 11133070
- DOI: 10.1016/s0960-894x(00)00558-8
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Solid-phase synthesis of 2,3-disubstituted indoles: discovery of a novel, high-affinity, selective h5-HT2A antagonist
Bioorg Med Chem Lett.
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Abstract
The application of a novel solid-phase synthesis of 2,3-disubstituted indoles utilizing a carbamate indole linker is described resulting in the identification of the novel, high-affinity, selective h5-HT2A antagonist 19.
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