Synthesis of Delta(1)-1,2-diazetines via a Diels-Alder cycloaddition approach
- PMID: 11574026
- DOI: 10.1021/ol0164942
Synthesis of Delta(1)-1,2-diazetines via a Diels-Alder cycloaddition approach
Abstract
[reaction: see text] A novel method for the synthesis of Delta(1)-1,2-diazetines is presented. Diels-Alder cycloaddition of dienophile 4 with five dienes afforded cycloadducts in good to excellent yields. Four of the obtained cycloadducts were converted to the corresponding diazetines.
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