Discodermolide/Dictyostatin hybrids: synthesis and biological evaluation
- PMID: 12465908
- DOI: 10.1021/ol026942l
Discodermolide/Dictyostatin hybrids: synthesis and biological evaluation
Erratum in
- Org Lett. 2003 Feb 20;(5)4:603.
Abstract
[structure: see text] Two hybrid analogues of discodermolide and dictyostatin (3, 26) have been designed and synthesized. These are the first macrocyclic analogues of discodermolide and biological activities were evaluated and compared with linear discodermolide analogues.
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