doi: 10.1016/j.bmcl.2005.05.081.
Glycosidase inhibition by 1-glycosyl-4-phenyl triazoles
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- PMID: 15979309
- DOI: 10.1016/j.bmcl.2005.05.081
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Glycosidase inhibition by 1-glycosyl-4-phenyl triazoles
Bioorg Med Chem Lett.
.
Abstract
1-Glycosyl-4-phenyl triazoles have been prepared via a copper-mediated [3+2] cycloaddition of glycosyl azides with phenylacetylene. These triazoles have been evaluated for their ability to inhibit the enzymatic activity of glycosidases.
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