Skip to main page content
U.S. flag

An official website of the United States government

Dot gov

The .gov means it’s official.
Federal government websites often end in .gov or .mil. Before sharing sensitive information, make sure you’re on a federal government site.

Https

The site is secure.
The https:// ensures that you are connecting to the official website and that any information you provide is encrypted and transmitted securely.

Access keys NCBI Homepage MyNCBI Homepage Main Content Main Navigation
. 2006 Jun 15;16(12):3233-7.
doi: 10.1016/j.bmcl.2006.03.047. Epub 2006 Apr 5.

Discovery of indole-containing tetracycles as a new scaffold for androgen receptor ligands

Xuqing Zhang  1 , Xiaojie Li, George F Allan, Amy Musto, Scott G Lundeen, Zhihua Sui
Affiliations

Discovery of indole-containing tetracycles as a new scaffold for androgen receptor ligands

Xuqing Zhang et al. Bioorg Med Chem Lett. .

Abstract

A novel series of tetracyclic indoles have been designed, synthesized and evaluated as androgen receptor (AR) ligands. Studies of structure-activity relationships (SARs) were investigated, which led to some compounds in this series as strong binders to androgen receptors.

PubMed Disclaimer

LinkOut - more resources