This site needs JavaScript to work properly. Please enable it to take advantage of the complete set of features!

Skip to main page content

Add to Collections

Your saved search

Name of saved search:

Search terms:

Test search terms

Would you like email updates of new search results?

Yes
No

Email: (change)

Frequency:

Which day?

Which day?

Report format:

Send at most:

Send even when there aren't any new results

Optional text in email:

Your RSS Feed

Review

. 1991 Nov;19(4):899-901.

doi: 10.1042/bst0190899.

Development of novel oestrogen-receptor antagonists

A E Wakeling¹, J Bowler

Affiliations

PMID: 1794580
DOI: 10.1042/bst0190899

Review

Development of novel oestrogen-receptor antagonists

A E Wakeling et al. Biochem Soc Trans. 1991 Nov.

. 1991 Nov;19(4):899-901.

doi: 10.1042/bst0190899.

Authors

A E Wakeling¹, J Bowler

Affiliation

¹ Research I, ICI Pharmaceuticals, Macclesfield, Cheshire, U.K.

PMID: 1794580
DOI: 10.1042/bst0190899

No abstract available

PubMed Disclaimer

Similar articles

Role of ligand in oestrogen-receptor function.
Parker MG, Fawell SE, Danielian P, Arbuckle N. Parker MG, et al. Biochem Soc Trans. 1991 Nov;19(4):897-9. doi: 10.1042/bst0190897. Biochem Soc Trans. 1991. PMID: 1794579 No abstract available.
Responses to pure antiestrogens (ICI 164384, ICI 182780) in estrogen-sensitive and -resistant experimental and clinical breast cancer.
Nicholson RI, Gee JM, Manning DL, Wakeling AE, Montano MM, Katzenellenbogen BS. Nicholson RI, et al. Ann N Y Acad Sci. 1995 Jun 12;761:148-63. doi: 10.1111/j.1749-6632.1995.tb31376.x. Ann N Y Acad Sci. 1995. PMID: 7625718 Review. No abstract available.
Estrogen induces death of tamoxifen-resistant MCF-7 cells: contrasting effect of the estrogen receptor downregulator fulvestrant.
Planas-Silva MD, Waltz PK, Kilker RL. Planas-Silva MD, et al. J Steroid Biochem Mol Biol. 2006 Mar;98(4-5):193-8. doi: 10.1016/j.jsbmb.2005.10.003. Epub 2006 Feb 7. J Steroid Biochem Mol Biol. 2006. PMID: 16464573
Response to specific anti-oestrogen (ICI182780) in tamoxifen-resistant breast cancer.
Dowsett M, Johnston SR, Iveson TJ, Smith IE. Dowsett M, et al. Lancet. 1995 Feb 25;345(8948):525. doi: 10.1016/s0140-6736(95)90624-x. Lancet. 1995. PMID: 7861903 Clinical Trial. No abstract available.
Pure antiestrogens and breast cancer.
Elkak AE, Mokbel K. Elkak AE, et al. Curr Med Res Opin. 2001;17(4):282-9. Curr Med Res Opin. 2001. PMID: 11922402 Review.

See all similar articles

Cited by

Estrogen Receptor-α Targeting: PROTACs, SNIPERs, Peptide-PROTACs, Antibody Conjugated PROTACs and SNIPERs.
Negi A, Kesari KK, Voisin-Chiret AS. Negi A, et al. Pharmaceutics. 2022 Nov 19;14(11):2523. doi: 10.3390/pharmaceutics14112523. Pharmaceutics. 2022. PMID: 36432713 Free PMC article. Review.
From Pure Antagonists to Pure Degraders of the Estrogen Receptor: Evolving Strategies for the Same Target.
Mottamal M, Kang B, Peng X, Wang G. Mottamal M, et al. ACS Omega. 2021 Mar 30;6(14):9334-9343. doi: 10.1021/acsomega.0c06362. eCollection 2021 Apr 13. ACS Omega. 2021. PMID: 33869913 Free PMC article. Review.
Jostling for position: optimizing linker location in the design of estrogen receptor-targeting PROTACs.
Cyrus K, Wehenkel M, Choi EY, Lee H, Swanson H, Kim KB. Cyrus K, et al. ChemMedChem. 2010 Jul 5;5(7):979-85. doi: 10.1002/cmdc.201000146. ChemMedChem. 2010. PMID: 20512796 Free PMC article.
Oestrogens and spermatogenesis.
Carreau S, Hess RA. Carreau S, et al. Philos Trans R Soc Lond B Biol Sci. 2010 May 27;365(1546):1517-35. doi: 10.1098/rstb.2009.0235. Philos Trans R Soc Lond B Biol Sci. 2010. PMID: 20403867 Free PMC article. Review.
Differential hormonal regulation of estrogen receptors ERalpha and ERbeta and androgen receptor expression in rat efferent ductules.
Oliveira CA, Mahecha GA, Carnes K, Prins GS, Saunders PT, França LR, Hess RA. Oliveira CA, et al. Reproduction. 2004 Jul;128(1):73-86. doi: 10.1530/rep.1.00136. Reproduction. 2004. PMID: 15232065 Free PMC article.

Publication types

Actions

MeSH terms

Actions
Actions
Actions
Actions
Actions
Actions
Actions
Actions
Actions
Actions
Actions
Actions
Actions
Actions
Actions

Substances

Actions
Actions
Actions
Actions
Actions
Actions
Actions

LinkOut - more resources

Full Text Sources
- Silverchair Information Systems
Other Literature Sources
- The Lens - Patent Citations Database