Developments in nonsteroidal antiandrogens targeting the androgen receptor
- PMID: 20853390
- DOI: 10.1002/cmdc.201000259
Developments in nonsteroidal antiandrogens targeting the androgen receptor
Similar articles
-
Synthesis and preliminary investigations into novel 1,2,3-triazole-derived androgen receptor antagonists inspired by bicalutamide.Bioorg Med Chem Lett. 2014 Nov 1;24(21):4948-53. doi: 10.1016/j.bmcl.2014.09.036. Epub 2014 Sep 19. Bioorg Med Chem Lett. 2014. PMID: 25301770
-
Circumventing anti-androgen resistance by molecular design.J Am Chem Soc. 2007 Apr 4;129(13):3822-3. doi: 10.1021/ja0701154. Epub 2007 Mar 10. J Am Chem Soc. 2007. PMID: 17348658 Free PMC article.
-
Synthesis and structure-activity relationships of the first ferrocenyl-aryl-hydantoin derivatives of the nonsteroidal antiandrogen nilutamide.J Med Chem. 2008 Mar 27;51(6):1791-9. doi: 10.1021/jm701264d. Epub 2008 Feb 28. J Med Chem. 2008. PMID: 18303829
-
Non-Steroidal Androgen Receptor Antagonists and Prostate Cancer: A Survey on Chemical Structures Binding this Fast-Mutating Target.Curr Med Chem. 2019;26(33):6053-6073. doi: 10.2174/0929867325666180913095239. Curr Med Chem. 2019. PMID: 30209993 Review.
-
'Casodex': defining the role of antiandrogens.Cancer J Sci Am. 1997 Jul-Aug;3(4):204-8. Cancer J Sci Am. 1997. PMID: 9263624 Review. No abstract available.
Cited by
-
An Aminosteroid Derivative Shows Higher In Vitro and In Vivo Potencies than Gold Standard Drugs in Androgen-Dependent Prostate Cancer Models.Cancers (Basel). 2023 Jun 2;15(11):3033. doi: 10.3390/cancers15113033. Cancers (Basel). 2023. PMID: 37296995 Free PMC article.
-
Revisiting the SAR of the Antischistosomal Aryl Hydantoin (Ro 13-3978).J Med Chem. 2016 Dec 8;59(23):10705-10718. doi: 10.1021/acs.jmedchem.6b01410. Epub 2016 Nov 28. J Med Chem. 2016. PMID: 27933964 Free PMC article.
-
One-Pot Multicomponent Synthesis of Methoxybenzo[h]quinoline-3-carbonitrile Derivatives; Anti-Chagas, X-ray, and In Silico ADME/Tox Profiling Studies.Molecules. 2021 Nov 19;26(22):6977. doi: 10.3390/molecules26226977. Molecules. 2021. PMID: 34834070 Free PMC article.
-
Methoxychalcone inhibitors of androgen receptor translocation and function.Bioorg Med Chem Lett. 2012 Mar 1;22(5):2105-9. doi: 10.1016/j.bmcl.2011.12.141. Epub 2012 Jan 21. Bioorg Med Chem Lett. 2012. PMID: 22310230 Free PMC article.
Publication types
MeSH terms
Substances
LinkOut - more resources
Full Text Sources
Other Literature Sources