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Editorial
. 2024 Jul;181(14):2091-2094.
doi: 10.1111/bph.16419. Epub 2024 May 26.

Highlights and hot topics in GPCR research from 'Down Under'

Nicola J Smith  1 , Lauren T May  2 , Natasha L Grimsey  3   4   5
Affiliations
Free article
Editorial

Highlights and hot topics in GPCR research from 'Down Under'

Nicola J Smith et al. Br J Pharmacol. 2024 Jul.
Free article

Abstract

This article is part of a themed issue Therapeutic Targeting of G Protein-Coupled Receptors: hot topics from the Australasian Society of Clinical and Experimental Pharmacologists and Toxicologists 2021 Virtual Annual Scientific Meeting. To view the other articles in this section visit http://onlinelibrary.wiley.com/doi/10.1111/bph.v181.14/issuetoc.

Keywords: G protein; G protein‐coupled receptors (GPCRs); PROTAC; allostery; artificial intelligence; cardiometabolic; cardiovascular; disease mechanisms; effectors; epilepsy; fibrosis; orphan; phosphoproteomics; regulation; schizophrenia; second messengers.

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References

REFERENCES

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    1. Carruthers, E. R., & Grimsey, N. L. (2024). Cannabinoid CB2 receptor orthologues; in vitro function and perspectives for preclinical to clinical translation. British Journal of Pharmacology, 181(14), 2247–2269. https://doi.org/10.1111/bph.16172
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