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Editorial
. 2024 Sep 12;67(17):14693-14696.
doi: 10.1021/acs.jmedchem.4c01721. Epub 2024 Aug 8.

Demystifying Functional Parameters for Irreversible Enzyme Inhibitors

David E Heppner  1 , Blessing C Ogboo  1 , Daniel A Urul  2 , Earl W May  2 , Erik M Schaefer  2 , Andrew S Murkin  1 , Matthias Gehringer  3
Affiliations
Editorial

Demystifying Functional Parameters for Irreversible Enzyme Inhibitors

David E Heppner et al. J Med Chem. .
No abstract available

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Figures

Figure 1.
Figure 1.
A one-slide summary of the mechanisms of reversible (1-step, non-covalent) and irreversible (2-step, covalent) enzyme inhibitors and accompanying functional parameters.
See this image and copyright information in PMC

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