Novel Isotryptamine Tetracycles as 5‑HT2A Agonists for Treating Brain Disorders
- PMID: 40529052
- PMCID: PMC12169452
- DOI: 10.1021/acsmedchemlett.5c00246
Novel Isotryptamine Tetracycles as 5‑HT2A Agonists for Treating Brain Disorders
Abstract
Provided herein are novel isotryptamine tetracycles as 5-HT2A agonists, pharmaceutical compositions, use of such compounds in treating brain disorders, and processes for preparing such compounds.
Published 2025 by American Chemical Society.
References
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- Cummins, B. R. ; Billac, G. B. ; Nichols, D. E. ; Nichols, C. D. . 5-HT2A receptors: Pharmacology and functional selectivity. Pharmacol. Rev. 2025, in press. 10.1016/j.pharmr.2025.100059. https://www.sciencedirect.com/science/article/pii/S0031699725074678 - DOI - PubMed
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