Novel Bicyclic Heterocycles as MRGPRX2 Antagonists for Treating Inflammatory Diseases
- PMID: 40529074
- PMCID: PMC12169468
- DOI: 10.1021/acsmedchemlett.5c00305
Novel Bicyclic Heterocycles as MRGPRX2 Antagonists for Treating Inflammatory Diseases
Abstract
Provided herein are novel bicyclic heterocycles as MRGPRX2 antagonists, pharmaceutical compositions, use of such compounds in treating inflammatory diseases, and processes for preparing such compounds.
Published 2025 by American Chemical Society.
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