doi: 10.1016/0014-2999(78)90031-6.
Influence of GABA receptor agonists and antagonists on the binding of 3H-diazepam to the benzodiazepine receptor
- PMID: 720385
- DOI: 10.1016/0014-2999(78)90031-6
Item in Clipboard
Influence of GABA receptor agonists and antagonists on the binding of 3H-diazepam to the benzodiazepine receptor
Eur J Pharmacol.
.
Abstract
The GABA receptor agonists, GABA and muscimol, increased, while the GABA receptor antagonist, (+)-bicuculline, decreased the affinity of the benzodiazepine receptor for 3H-diazepam. The effect was seen at both 0 and 25 degrees C in spite of a large difference of affinity for 3H-diazepam at the two temperatures.
Similar articles
-
Partial agonists for brain GABA/benzodiazepine receptor complex.Nature. 1979 Jul 26;280(5720):331-3. doi: 10.1038/280331a0. Nature. 1979. PMID: 460407 No abstract available.
-
Stimulation of benzodiazepine receptor binding by gamma-aminobutyric acid.Proc Natl Acad Sci U S A. 1979 Feb;76(2):1004-6. doi: 10.1073/pnas.76.2.1004. Proc Natl Acad Sci U S A. 1979. PMID: 284378 Free PMC article.
-
Two or more conformations of benzodiazepine receptors depending on GABA receptors and other variables.Adv Biochem Psychopharmacol. 1980;21:301-12. Adv Biochem Psychopharmacol. 1980. PMID: 6246746 No abstract available.
-
GABA-benzodiazepine interactions: physiological, pharmacological and developmental aspects.Fed Proc. 1980 Oct;39(12):3043-9. Fed Proc. 1980. PMID: 6252066 Review.
-
The benzodiazepine receptor of mammalian brain.Fed Proc. 1980 Oct;39(12):3032-8. Fed Proc. 1980. PMID: 6998742 Review.
Cited by
-
Effects of valproate on hyponeophagia in rats: competitive antagonism with picrotoxin and non-competitive antagonism with RO 15-1788.Psychopharmacology (Berl). 1985;86(3):313-7. doi: 10.1007/BF00432220. Psychopharmacology (Berl). 1985. PMID: 2994145
-
The GABA postsynaptic membrane receptor-ionophore complex. Site of action of convulsant and anticonvulsant drugs.Mol Cell Biochem. 1981 Sep 25;39:261-79. doi: 10.1007/BF00232579. Mol Cell Biochem. 1981. PMID: 6273709 Review.
-
Evaluating chemical effects on human neural cells through calcium imaging and deep learning.iScience. 2024 Nov 1;27(12):111298. doi: 10.1016/j.isci.2024.111298. eCollection 2024 Dec 20. iScience. 2024. PMID: 39634567 Free PMC article.
-
gamma-Aminobutyric acid and benzodiazepine receptors: copurification and characterization.Proc Natl Acad Sci U S A. 1981 Mar;78(3):1939-42. doi: 10.1073/pnas.78.3.1939. Proc Natl Acad Sci U S A. 1981. PMID: 6112752 Free PMC article.
-
Methylmercury modulates GABAA receptor complex differentially in rat cortical and cerebellar membranes in vitro.Neurochem Res. 1995 Jun;20(6):659-62. doi: 10.1007/BF01705532. Neurochem Res. 1995. PMID: 7566360
MeSH terms
Substances
LinkOut - more resources
Full Text Sources
