Besson T - Search Results

1

Design and synthesis of thiazolo[5,4-f]quinazolines as DYRK1A inhibitors, part II.

Foucourt A, Hédou D, Dubouilh-Benard C, Girard A, Taverne T, Casagrande AS, Désiré L, Leblond B, Besson T. Foucourt A, et al. Among authors: besson t. Molecules. 2014 Sep 26;19(10):15411-39. doi: 10.3390/molecules191015411. Molecules. 2014. PMID: 25264830 Free PMC article.

2

Dissociation reactions of free tetrapyridinium tetracations and of their catenanes.

Roithová J, Milko P, Ricketts CL, Schröder D, Besson T, Dekoj V, Belohradský M. Roithová J, et al. Among authors: besson t. J Am Chem Soc. 2007 Aug 22;129(33):10141-8. doi: 10.1021/ja071058h. Epub 2007 Jul 26. J Am Chem Soc. 2007. PMID: 17655231

3

Microwave-assisted synthesis of bioactive quinazolines and quinazolinones.

Besson T, Chosson E. Besson T, et al. Comb Chem High Throughput Screen. 2007 Dec;10(10):903-17. doi: 10.2174/138620707783220356. Comb Chem High Throughput Screen. 2007. PMID: 18288950 Review.

4

Synthesis and biological evaluation of N-arylbenzo[b]thieno[3,2-d]pyrimidin-4-amines and their pyrido and pyrazino analogues as Ser/Thr kinase inhibitors.

Loidreau Y, Marchand P, Dubouilh-Benard C, Nourrisson MR, Duflos M, Lozach O, Loaëc N, Meijer L, Besson T. Loidreau Y, et al. Among authors: besson t. Eur J Med Chem. 2012 Dec;58:171-83. doi: 10.1016/j.ejmech.2012.10.006. Epub 2012 Oct 16. Eur J Med Chem. 2012. PMID: 23124214

5

Synthesis and biological evaluation of N-aryl-7-methoxybenzo[b]furo[3,2-d]pyrimidin-4-amines and their N-arylbenzo[b]thieno[3,2-d]pyrimidin-4-amine analogues as dual inhibitors of CLK1 and DYRK1A kinases.

Loidreau Y, Marchand P, Dubouilh-Benard C, Nourrisson MR, Duflos M, Loaëc N, Meijer L, Besson T. Loidreau Y, et al. Among authors: besson t. Eur J Med Chem. 2013 Jan;59:283-95. doi: 10.1016/j.ejmech.2012.11.030. Epub 2012 Nov 24. Eur J Med Chem. 2013. PMID: 23237976

6

Synthesis of novel 7-substituted pyrido[2',3':4,5]furo[3,2-d]pyrimidin-4-amines and their N-aryl analogues and evaluation of their inhibitory activity against Ser/Thr kinases.

Deau E, Loidreau Y, Marchand P, Nourrisson MR, Loaëc N, Meijer L, Levacher V, Besson T. Deau E, et al. Among authors: besson t. Bioorg Med Chem Lett. 2013 Dec 15;23(24):6784-8. doi: 10.1016/j.bmcl.2013.10.019. Epub 2013 Oct 17. Bioorg Med Chem Lett. 2013. PMID: 24176400

7

Discovery of a novel broad-spectrum antifungal agent derived from albaconazole.

Guillon R, Pagniez F, Picot C, Hédou D, Tonnerre A, Chosson E, Duflos M, Besson T, Logé C, Le Pape P. Guillon R, et al. Among authors: besson t. ACS Med Chem Lett. 2013 Jan 17;4(2):288-92. doi: 10.1021/ml300429p. eCollection 2013 Feb 14. ACS Med Chem Lett. 2013. PMID: 24900660 Free PMC article.

8

Design and synthesis of thiazolo[5,4-f]quinazolines as DYRK1A inhibitors, part I.

Foucourt A, Hédou D, Dubouilh-Benard C, Désiré L, Casagrande AS, Leblond B, Loäec N, Meijer L, Besson T. Foucourt A, et al. Among authors: besson t. Molecules. 2014 Sep 29;19(10):15546-71. doi: 10.3390/molecules191015546. Molecules. 2014. PMID: 25268714 Free PMC article.

9

Synthesis and molecular modelling studies of 8-arylpyrido[3',2':4,5]thieno[3,2-d]pyrimidin-4-amines as multitarget Ser/Thr kinases inhibitors.

Loidreau Y, Deau E, Marchand P, Nourrisson MR, Logé C, Coadou G, Loaëc N, Meijer L, Besson T. Loidreau Y, et al. Among authors: besson t. Eur J Med Chem. 2015 Mar 6;92:124-34. doi: 10.1016/j.ejmech.2014.12.038. Epub 2014 Dec 23. Eur J Med Chem. 2015. PMID: 25549552

10

A novel DYRK1A (dual specificity tyrosine phosphorylation-regulated kinase 1A) inhibitor for the treatment of Alzheimer's disease: effect on Tau and amyloid pathologies in vitro.

Coutadeur S, Benyamine H, Delalonde L, de Oliveira C, Leblond B, Foucourt A, Besson T, Casagrande AS, Taverne T, Girard A, Pando MP, Désiré L. Coutadeur S, et al. Among authors: besson t. J Neurochem. 2015 May;133(3):440-51. doi: 10.1111/jnc.13018. Epub 2015 Jan 26. J Neurochem. 2015. PMID: 25556849 Free article.

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