Validation, Key Pharmacophores, and X-ray Cocrystal Structures of Novel Biochemically and Cellularly Active WRN Inhibitors Derived from a DNA-Encoded Library Screen.
Tong Y, Baker KA, Chapman AM, Elsen NL, Fowler F, George MD, Gesmundo NJ, Hatton H, Hickey M, Hutchins CW, Jeffries CL, Kelly A, Korepanova A, Miller IR, Nocek B, Panchal SC, Pemberton OA, Qiu W, Talaty NN, Hin Tang HY, Towne D, Zhang M, Zhao Y, Gopalakrishnan SM, Sun C, Kort ME, Dart MJ, Firestone AJ.
Tong Y, et al. Among authors: gopalakrishnan sm.
J Med Chem. 2025 Jun 26;68(12):12434-12456. doi: 10.1021/acs.jmedchem.4c03029. Epub 2025 Jun 5.
J Med Chem. 2025.
PMID: 40472162