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Tissue-specific regulation of gene expression via unproductive splicing.
Mironov A, Petrova M, Margasyuk S, Vlasenok M, Mironov AA, Skvortsov D, Pervouchine DD. Mironov A, et al. Among authors: skvortsov d. Nucleic Acids Res. 2023 Apr 24;51(7):3055-3066. doi: 10.1093/nar/gkad161. Nucleic Acids Res. 2023. PMID: 36912101 Free PMC article.
Electrochemical Detection of a Novel Pt(IV) Prodrug with the Metronidazole Axial Ligand in the Hypoxic Area.
Spector DV, Erofeev AS, Gorelkin PV, Vaneev AN, Akasov RA, Ul'yanovskiy NV, Nikitina VN, Semkina AS, Vlasova KY, Soldatov MA, Trigub AL, Skvortsov DA, Finko AV, Zyk NV, Sakharov DA, Majouga AG, Beloglazkina EK, Krasnovskaya OO. Spector DV, et al. Inorg Chem. 2022 Sep 19;61(37):14705-14717. doi: 10.1021/acs.inorgchem.2c02062. Epub 2022 Sep 1. Inorg Chem. 2022. PMID: 36047922
Biotinylated Pt(IV) prodrugs with elevated lipophilicity and cytotoxicity.
Spector D, Erofeev A, Gorelkin P, Skvortsov D, Trigub A, Markova A, Nikitina V, Ul'yanovskiy N, Shtil' A, Semkina A, Vlasova K, Zyk N, Majouga A, Beloglazkina E, Krasnovskaya O. Spector D, et al. Among authors: skvortsov d. Dalton Trans. 2023 Jan 24;52(4):866-871. doi: 10.1039/d2dt03662b. Dalton Trans. 2023. PMID: 36629146
Mixed valence copper(I,II) binuclear complexes with unexpected structure: synthesis, biological properties and anticancer activity.
Majouga AG, Zvereva MI, Rubtsova MP, Skvortsov DA, Mironov AV, Azhibek DM, Krasnovskaya OO, Gerasimov VM, Udina AV, Vorozhtsov NI, Beloglazkina EK, Agron L, Mikhina LV, Tretyakova AV, Zyk NV, Zefirov NS, Kabanov AV, Dontsova OA. Majouga AG, et al. J Med Chem. 2014 Jul 24;57(14):6252-8. doi: 10.1021/jm500154f. Epub 2014 Jul 8. J Med Chem. 2014. PMID: 24950478
PSMA-targeted small-molecule docetaxel conjugate: Synthesis and preclinical evaluation.
Machulkin AE, Uspenskaya AA, Zyk NY, Nimenko EA, Ber AP, Petrov SA, Shafikov RR, Skvortsov DA, Smirnova GB, Borisova YA, Pokrovsky VS, Kolmogorov VS, Vaneev AN, Ivanenkov YA, Khudyakov AD, Kovalev SV, Erofeev AS, Gorelkin PV, Beloglazkina EK, Zyk NV, Khazanova ES, Majouga AG. Machulkin AE, et al. Among authors: skvortsov da. Eur J Med Chem. 2022 Jan 5;227:113936. doi: 10.1016/j.ejmech.2021.113936. Epub 2021 Oct 23. Eur J Med Chem. 2022. PMID: 34717125
Synthesis and Biological Evaluation of PSMA Ligands with Aromatic Residues and Fluorescent Conjugates Based on Them.
Machulkin AE, Shafikov RR, Uspenskaya AA, Petrov SA, Ber AP, Skvortsov DA, Nimenko EA, Zyk NU, Smirnova GB, Pokrovsky VS, Abakumov MA, Saltykova IV, Akhmirov RT, Garanina AS, Polshakov VI, Saveliev OY, Ivanenkov YA, Aladinskaya AV, Finko AV, Yamansarov EU, Krasnovskaya OO, Erofeev AS, Gorelkin PV, Dontsova OA, Beloglazkina EK, Zyk NV, Khazanova ES, Majouga AG. Machulkin AE, et al. J Med Chem. 2021 Apr 22;64(8):4532-4552. doi: 10.1021/acs.jmedchem.0c01935. Epub 2021 Apr 6. J Med Chem. 2021. PMID: 33822606
138 results