Besson T - Search Results

1

DYRK1A inhibition results in MYC and ERK activation rendering KMT2A-R acute lymphoblastic leukemia cells sensitive to BCL2 inhibition.

Ayyadevara VSSA, Wertheim G, Gaur S, Chukinas JA, Loftus JP, Lee SJ, Kumar A, Swaminathan S, Bhansali RS, Childers W, Geng H, Milne TA, Hua X, Bernt KM, Besson T, Shi J, Crispino JD, Carroll M, Tasian SK, Hurtz C. Ayyadevara VSSA, et al. Among authors: besson t. Leukemia. 2025 May;39(5):1078-1089. doi: 10.1038/s41375-025-02575-w. Epub 2025 Mar 27. Leukemia. 2025. PMID: 40148558 Free PMC article.

2

Review on the Synthesis and Therapeutic Potential of Pyrido[2,3-d], [3,2-d], [3,4-d] and [4,3-d]pyrimidine Derivatives.

Campos JF, Besson T, Berteina-Raboin S. Campos JF, et al. Among authors: besson t. Pharmaceuticals (Basel). 2022 Mar 14;15(3):352. doi: 10.3390/ph15030352. Pharmaceuticals (Basel). 2022. PMID: 35337149 Free PMC article. Review.

3

Synthesis of Bioactive 2-(Arylamino)thiazolo[5,4-f]-quinazolin-9-ones via the Hügershoff Reaction or Cu- Catalyzed Intramolecular C-S Bond Formation.

Hédou D, Dubouilh-Benard C, Loaëc N, Meijer L, Fruit C, Besson T. Hédou D, et al. Among authors: besson t. Molecules. 2016 Jun 18;21(6):794. doi: 10.3390/molecules21060794. Molecules. 2016. PMID: 27322235 Free PMC article.

4

Synthesis of Thiazolo[5,4-f]quinazolin-9(8H)-ones as Multi-Target Directed Ligands of Ser/Thr Kinases.

Hédou D, Godeau J, Loaëc N, Meijer L, Fruit C, Besson T. Hédou D, et al. Among authors: besson t. Molecules. 2016 Apr 30;21(5):578. doi: 10.3390/molecules21050578. Molecules. 2016. PMID: 27144552 Free PMC article.

5

Demonstration of Green Solvent Performance on O,S,N-Heterocycles Synthesis: Metal-Free Click Chemistry and Buchwald-Hartwig Coupling.

Campos JF, Cailler M, Claudel R, Prot B, Besson T, Berteina-Raboin S. Campos JF, et al. Among authors: besson t. Molecules. 2021 Feb 18;26(4):1074. doi: 10.3390/molecules26041074. Molecules. 2021. PMID: 33670633 Free PMC article.

6

Synthesis of 2-Mercapto-(2-Oxoindolin-3-Ylidene)Acetonitriles from 3-(4-Chloro-5H-1,2,3-Dithiazol-5-Ylidene)Indolin-2-ones.

Letribot B, Delatouche R, Rouillard H, Bonnet A, Chérouvrier JR, Domon L, Besson T, Thiéry V. Letribot B, et al. Among authors: besson t. Molecules. 2018 Jun 8;23(6):1390. doi: 10.3390/molecules23061390. Molecules. 2018. PMID: 29890669 Free PMC article.

7

An Unusual Binding Model of the Methyl 9-Anilinothiazolo[5,4-f] quinazoline-2-carbimidates (EHT 1610 and EHT 5372) Confers High Selectivity for Dual-Specificity Tyrosine Phosphorylation-Regulated Kinases.

Chaikuad A, Diharce J, Schröder M, Foucourt A, Leblond B, Casagrande AS, Désiré L, Bonnet P, Knapp S, Besson T. Chaikuad A, et al. Among authors: besson t. J Med Chem. 2016 Nov 23;59(22):10315-10321. doi: 10.1021/acs.jmedchem.6b01083. Epub 2016 Nov 2. J Med Chem. 2016. PMID: 27766861

8

Microwave-Assisted Synthesis of Potential Bioactive Benzo-, Pyrido- or Pyrazino-thieno[3,2-d]pyrimidin-4-amine Analogs of MPC-6827.

Loidreau Y, Nourrisson MR, Fruit C, Corbière C, Marchand P, Besson T. Loidreau Y, et al. Among authors: besson t. Pharmaceuticals (Basel). 2020 Aug 19;13(9):202. doi: 10.3390/ph13090202. Pharmaceuticals (Basel). 2020. PMID: 32825171 Free PMC article.

9

26th Annual GP2A Medicinal Chemistry Conference & 32nd Journées Franco-Belges de Pharmacochimie.

Dallemagne P, Rochais C, Marchand P, Besson T. Dallemagne P, et al. Among authors: besson t. Pharmaceuticals (Basel). 2019 May 16;12(2):73. doi: 10.3390/ph12020073. Pharmaceuticals (Basel). 2019. PMID: 31100957 Free PMC article.

10

A skills framework integrating professionally relevant medicinal chemistry proficiencies to strengthen the contemporary practice of pharmacy.

Decombat C, Duval O, Besson T, Bourel L, Pudlo M. Decombat C, et al. Among authors: besson t. Ann Pharm Fr. 2022 Mar;80(2):176-186. doi: 10.1016/j.pharma.2021.07.001. Epub 2021 Jul 24. Ann Pharm Fr. 2022. PMID: 34314680 Review.

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