Optimization and Characterization of N-Acetamide Indoles as Antimalarials That Target PfATP4.
Awalt JK, Ooi ZK, Ashton TD, Mansouri M, Calic PPS, Zhou Q, Vasanthan S, Lee S, Loi K, Jarman KE, Penington JS, Qiu D, Zhang X, Lehane AM, Mao EY, Gancheva MR, Wilson DW, Giannangelo C, MacRaild CA, Creek DJ, Yeo T, Sheth T, Fidock DA, Churchyard A, Baum J, Famodimu MT, Delves MJ, Kristan M, Stewart L, Sutherland CJ, Coyle R, Jagoe H, Lee MCS, Chowdury M, de Koning-Ward TF, Baud D, Brand S, Jackson PF, Cowman AF, Dans MG, Sleebs BE.
Awalt JK, et al. Among authors: penington js.
J Med Chem. 2025 Apr 24;68(8):8933-8966. doi: 10.1021/acs.jmedchem.5c00614. Epub 2025 Apr 14.
J Med Chem. 2025.
PMID: 40228810
Free PMC article.