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Page 1
Weinreb Amides as Directing Groups for Transition Metal-Catalyzed C-H Functionalizations.
Kalepu J, Pilarski LT. Kalepu J, et al. Molecules. 2019 Feb 26;24(5):830. doi: 10.3390/molecules24050830. Molecules. 2019. PMID: 30813564 Free PMC article. Review.
Weinreb amides are a privileged, multi-functional group with well-established utility in classical synthesis. Recently, several studies have demonstrated the use of Weinreb amides as interesting substrates in transition metal-catalyzed C-H functionalization reaction …
Weinreb amides are a privileged, multi-functional group with well-established utility in classical synthesis. Recently, several studi …
Weinreb Amide Approach to the Practical Synthesis of a Key Remdesivir Intermediate.
Xie Y, Hu T, Zhang Y, Wei D, Zheng W, Zhu F, Tian G, Aisa HA, Shen J. Xie Y, et al. J Org Chem. 2021 Apr 2;86(7):5065-5072. doi: 10.1021/acs.joc.0c02986. Epub 2021 Mar 18. J Org Chem. 2021. PMID: 33733767
Adequate supplies of remdesivir are highly warranted to cope with this global public health crisis. Herein, we report a Weinreb amide approach for preparing the key intermediate of remdesivir in the glycosylation step where overaddition side reactions are eliminated. Start …
Adequate supplies of remdesivir are highly warranted to cope with this global public health crisis. Herein, we report a Weinreb amide …
Acromegaly.
Weinreb J, Arora S. Weinreb J, et al. N Engl J Med. 2023 Jan 5;388(1):70. doi: 10.1056/NEJMicm2205570. N Engl J Med. 2023. PMID: 36599064 No abstract available.
PI-RADS Prostate Imaging - Reporting and Data System: 2015, Version 2.
Weinreb JC, Barentsz JO, Choyke PL, Cornud F, Haider MA, Macura KJ, Margolis D, Schnall MD, Shtern F, Tempany CM, Thoeny HC, Verma S. Weinreb JC, et al. Eur Urol. 2016 Jan;69(1):16-40. doi: 10.1016/j.eururo.2015.08.052. Epub 2015 Oct 1. Eur Urol. 2016. PMID: 26427566 Free PMC article.
Author Reply.
Syed JS, Lu A, Nguyen KA, Sprenkle PC, Weinreb JC. Syed JS, et al. Urology. 2017 Jul;105:122. doi: 10.1016/j.urology.2017.01.050. Epub 2017 Apr 24. Urology. 2017. PMID: 28449978 No abstract available.
Acid-Enabled Palladium-Catalyzed beta-C(sp(3))-H Functionalization of Weinreb Amides.
Yang L, Xie H, An G, Li G. Yang L, et al. J Org Chem. 2021 Jun 4;86(11):7872-7880. doi: 10.1021/acs.joc.1c00781. Epub 2021 May 13. J Org Chem. 2021. PMID: 33985328
Herein, we report Pd(II)-catalyzed C(sp(3))-H arylation and alkenylation of Weinreb amides. A commercially available, inexpensive sulfonic acid was employed to enhance the coordination of the catalyst with weak-coordinating substrates by increasing the electrophilicity of …
Herein, we report Pd(II)-catalyzed C(sp(3))-H arylation and alkenylation of Weinreb amides. A commercially available, inexpensive sul …
Ligand-Enabled, Palladium-Catalyzed beta-C(sp(3))-H Arylation of Weinreb Amides.
Park H, Chekshin N, Shen PX, Yu JQ. Park H, et al. ACS Catal. 2018 Oct 5;8(10):9292-9297. doi: 10.1021/acscatal.8b03014. Epub 2018 Sep 5. ACS Catal. 2018. PMID: 31223513 Free PMC article.
We report the development of Pd(II)-catalyzed C(sp(3))-H arylation of Weinreb amides. This work demonstrates the first example of using Weinreb amide as a directing group for transition metal-catalyzed C(sp(3))-H activation. Both the inductive effect and the potenti …
We report the development of Pd(II)-catalyzed C(sp(3))-H arylation of Weinreb amides. This work demonstrates the first example of usi …
Synthesis of Weinreb amides using diboronic acid anhydride-catalyzed dehydrative amidation of carboxylic acids.
Shimada N , Takahashi N , Ohse N , Koshizuka M , Makino K . Shimada N , et al. Chem Commun (Camb). 2020 Nov 7;56(86):13145-13148. doi: 10.1039/d0cc05630h. Epub 2020 Oct 2. Chem Commun (Camb). 2020. PMID: 33007055
The first successful example of the direct synthesis of Weinreb amides using catalytic hydroxy-directed dehydrative amidation of carboxylic acids using the diboronic acid anhydride catalyst is described. ...
The first successful example of the direct synthesis of Weinreb amides using catalytic hydroxy-directed dehydrative amidation of carb …
Weinreb Amide, Ketone and Amine as Potential and Competitive Secondary Molecular Stations for Dibenzo-[24]Crown-8 in [2]Rotaxane Molecular Shuttles.
Gauthier M, Coutrot F. Gauthier M, et al. Chemistry. 2021 Dec 15;27(70):17576-17580. doi: 10.1002/chem.202103805. Epub 2021 Nov 24. Chemistry. 2021. PMID: 34738683
This paper reports the synthesis and study of new pH-sensitive DB24C8-based [2]rotaxane molecular shuttles that contain within their axle four potential sites of interaction for the DB24C8: ammonium, amine, Weinreb amide, and ketone. In the protonated state, the DB24C8 lay …
This paper reports the synthesis and study of new pH-sensitive DB24C8-based [2]rotaxane molecular shuttles that contain within their axle fo …
Reply.
Akagi T, Zangwill LM, Weinreb RN. Akagi T, et al. Ophthalmology. 2018 Mar;125(3):e22-e23. doi: 10.1016/j.ophtha.2017.10.013. Ophthalmology. 2018. PMID: 29458837 No abstract available.
2,870 results